KO

원료의약품

Sitagliptin Phosphate (시타글립틴인산염)

KDMF APIs

Sitagliptin Phosphate

Sitagliptin Phosphate 기본 정보

품목명 (한글)

시타글립틴인산염

분류

기타의 대사성 의약품

CAS No.

654671-78-0

KDMF 등록번호

수5217-4-ND

제조원

Mylan Laboratories Limited(Unit-1)

규격

In-house

품목 정보

Sitagliptin Phosphate 품목 정보

IUPAC Name

(3R)-3-amino-1-[3-(trifluoromethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one

Synonyms

Sitagliptin

Description

Sitagliptin is an oral dipeptidyl peptidase-4 (DPP-4) inhibitor used in conjunction with diet and exercise to improve glycemic control in patients with type 2 diabetes mellitus. The effect of this medication leads to glucose dependent increases in insulin and decreases in glucagon to improve control of blood sugar. Sitagliptin was granted FDA approval on October 16, 2006.

Certificate of Analysis

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