CN

原料药

Sitagliptin Phosphate

KDMF APIs

Sitagliptin Phosphate

Sitagliptin Phosphate 基本信息

韩文名称

시타글립틴인산염

分类

其他代谢类药物

CAS No.

654671-78-0

KDMF 登记号

수5217-4-ND

生产厂商

Mylan Laboratories Limited(Unit-1)

规格

In-house

品目信息

Sitagliptin Phosphate 品目信息

IUPAC Name

(3R)-3-amino-1-[3-(trifluoromethyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl]-4-(2,4,5-trifluorophenyl)butan-1-one

Synonyms

Sitagliptin

Description

Sitagliptin is an oral dipeptidyl peptidase-4 (DPP-4) inhibitor used in conjunction with diet and exercise to improve glycemic control in patients with type 2 diabetes mellitus. The effect of this medication leads to glucose dependent increases in insulin and decreases in glucagon to improve control of blood sugar. Sitagliptin was granted FDA approval on October 16, 2006.

Certificate of Analysis

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